Rhodium-Catalyzed Amidation of the Cage B(4)-H Bond in o-Carboranes with Dioxazolones by Carboxylic Acid-Assisted B(4)-H Bond Activation

  • Baek, Yonghyeon
  • Kim, Suhui
  • Son, Jeong-Yu
  • Lee, Kooyeon
  • Kim, Dongwook
  • 외 1명
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초록

A rhodium-catalyzed direct and regioselective amidation of the cage B(4)-H bond in a wide range of o-carboranes with alkyl-, aryl-, and heteroaryl-substituted dioxazolones is demonstrated by carboxylic acid-assisted B(4)-H bond activation in carborane clusters, providing a number of amidated o-carboranes in high yields with the release of carbon dioxide. Moreover, the selective 2-fold decarboxylative amidation reaction of the cage B(4)-H bond in o-carborane was accessed.

키워드

B-H activationrhodiumo-carboranedioxazoloneamidationC-H AMIDATIONNEUTRON-CAPTURE THERAPYB-HDRUG DISCOVERYBORONCHEMISTRYPHARMACOPHORESAZOBENZENESROUTE
제목
Rhodium-Catalyzed Amidation of the Cage B(4)-H Bond in o-Carboranes with Dioxazolones by Carboxylic Acid-Assisted B(4)-H Bond Activation
저자
Baek, YonghyeonKim, SuhuiSon, Jeong-YuLee, KooyeonKim, DongwookLee, Phil Ho
DOI
10.1021/acscatal.9b03380
발행일
2019-11
유형
Article
저널명
ACS Catalysis
9
11
페이지
10418 ~ 10425