γ-Selective allylic substitution reaction with Grignard reagents catalyzed by copper N-heterocyclic carbene complexes and its application to enantioselective synthesis

  • Tominaga, Satoshi
  • Oi, Yukinao
  • Kato, Toshio
  • An, Dukkeun
  • Okamoto, Sentaro
Citations

SCOPUS

112

초록

The reaction of allylic compounds with alkyl Grignard reagents in the presence of a catalytic amount of copper N-heterocyclic carbene (NHC) complexes proceeded predominantly in an S<inf>N</inf>2′ reaction pathway to give γ-substituted product in excellent yield. The method was applied to asymmetric reaction by using optically active NHC ligands. © 2004 Elsevier Ltd. All rights reserved.

키워드

Allylic substitutionAsymmetric reactionN-Heterocyclic carbeneOrganocopper
제목
γ-Selective allylic substitution reaction with Grignard reagents catalyzed by copper N-heterocyclic carbene complexes and its application to enantioselective synthesis
저자
Tominaga, SatoshiOi, YukinaoKato, ToshioAn, DukkeunOkamoto, Sentaro
DOI
10.1016/j.tetlet.2004.05.135
발행일
2004
유형
Article
저널명
Tetrahedron Letters
45
29
페이지
5585 ~ 5588