CONCISE SUBSTRATE-CONTROLLED ASYMMETRIC TOTAL SYNTHESIS OF (+)-3-(Z)-DIHYDRORHODOPHYTIN

  • Kim, Byungsook
  • Sohn, Te-ik
  • Kim, Sanghee
  • Kim, Deukjoon
  • Lee, Jongkook
Citations

WEB OF SCIENCE

11
Citations

SCOPUS

13

초록

The first asymmetric total synthesis of (+)-3-(Z)-dihydrorhodophytin (1) has been accomplished in 15 steps in 17% overall yield from readily available starting material 6 in a substrate-controlled manner. Key steps in our synthesis are a highly stereoselective dianion alkylation for the synthesis of the alpha,alpha'-anti-RCM substrate and a strategy for the introduction of the chlorine function.

키워드

Total Synthesis(+)-3-(Z)-DihydrorhodophytinIntermolecular Amide Enolate AlkylationRing-Closing MetathesisMedium-Sized OxacycleENANTIOSELECTIVE TOTAL-SYNTHESISSTRATEGY(+)-LAURENYNEALKYLATIONOXIDATION
제목
CONCISE SUBSTRATE-CONTROLLED ASYMMETRIC TOTAL SYNTHESIS OF (+)-3-(Z)-DIHYDRORHODOPHYTIN
저자
Kim, ByungsookSohn, Te-ikKim, SangheeKim, DeukjoonLee, Jongkook
DOI
10.3987/COM-10-S(E)76
발행일
2011-03-01
유형
Article
저널명
Heterocycles
82
2
페이지
1113 ~ +